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PU-H71 HCl
CAS No. 2095432-24-7
PU-H71 HCl ( —— )
产品货号. M36291 CAS No. 2095432-24-7
PU-H71 HCl (Zelavespib HCl) is a novel Hsp90 inhibitor, a novel purine-based analog, and a radiosensitizer that may be a promising agent for CIRT. PU-H71 HCL shows antitumor activity in many preclinical models of malignancy. PU-H71 HCL has an inhibitory effect on the protein expression levels of Rad51 and Ku70, which may be associated with the double chain break repair in the homologous recombination pathway and non-homologous end-joining pathway.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥2519 | 有现货 |
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| 5MG | ￥3472 | 有现货 |
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| 10MG | ￥5136 | 有现货 |
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| 25MG | ￥7718 | 有现货 |
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| 50MG | ￥10635 | 有现货 |
|
| 100MG | ￥14000 | 有现货 |
|
| 500MG | ￥28152 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称PU-H71 HCl
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述PU-H71 HCl (Zelavespib HCl) is a novel Hsp90 inhibitor, a novel purine-based analog, and a radiosensitizer that may be a promising agent for CIRT. PU-H71 HCL shows antitumor activity in many preclinical models of malignancy. PU-H71 HCL has an inhibitory effect on the protein expression levels of Rad51 and Ku70, which may be associated with the double chain break repair in the homologous recombination pathway and non-homologous end-joining pathway.
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产品描述PU-H71 HCl (Zelavespib HCl) is a novel Hsp90 inhibitor, a novel purine-based analog, and a radiosensitizer that may be a promising agent for CIRT. PU-H71 HCL shows antitumor activity in many preclinical models of malignancy. PU-H71 HCL has an inhibitory effect on the protein expression levels of Rad51 and Ku70, which may be associated with the double chain break repair in the homologous recombination pathway and non-homologous end-joining pathway.
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体外实验——
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体内实验——
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同义词——
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通路Cytoskeleton/Cell Adhesion Molecules
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靶点HSP
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受体HSP | DNA/RNA Synthesis
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研究领域——
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适应症——
化学信息
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CAS Number2095432-24-7
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分子量548.83
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分子式C18H22ClIN6O2S
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纯度>98% (HPLC)
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溶解度——
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SMILESCl.IC=1C=C2OCOC2=CC1SC3=NC=4C(=NC=NC4N3CCCNC(C)C)N
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
产品手册
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